Azelaprag free base · Synonyms: AMG-986 | AMG 986

Azelaprag is a candidate active molecule for an Apelin receptor agonist.

For research use only. Not for human or veterinary use.

Target Apelin Receptor (APJ)

Research area Others

Purity >98% Stock Inquire

Data Sheet SDS COA

Azelaprag structure

CAS No.: 2049980-18-7

Pack sizes & pricing

Size	Price	SKU	Stock
100 mg	USD 598.00	BP-01563-100mg	In stock	Get quote
250 mg	USD 825.00	BP-01563-250mg	In stock	Get quote
500 mg	USD 1,450.00	BP-01563-500mg	In stock	Get quote
1 g	USD 2,450.00	BP-01563-1g	In stock	Get quote
2 g	USD 3,920.00	BP-01563-2g	In stock	Get quote
5 g	Inquire	BP-01563-5g	In stock	Inquire

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Azelaprag (Example 263.0) is a candidate active molecule for an Apelin receptor agonist with an EC50 of 0.32 nM for the apelin receptor .

Azelaprag (Example 263.0) is an apelin receptor agonist agent candidate.

SMILES: N(S([C@H]([C@H](C)C=1N=CC(C)=CN1)C)(=O)=O)C=2N(C(=NN2)C=3C=C(C)C=NC3)C4=C(OC)C=CC=C4OC
InChIKey: DOMQFIFVDIAOOT-ROUUACIJSA-N

MW (average): 523.6070
Formula: C₂₅H₂₉N₇O₄S
CAS No.: 2049980-18-7
Physical state: Solid
Color: white to light yellow
Shipping: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage: Powder: 4℃, 2 years; In solvent: -20℃, 1 month

soluble in DMSO

[1]. WO2016187308A1.

[2]. Ason B, et.al. Cardiovascular response to small-molecule APJ activation. JCI Insight. 2020 Apr 23;5(8):e132898.

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