BiochemProbe — Life Science Research Reagents

Gilmelisib free base

Gilmelisib is an antineoplastic.

For research use only. Not for human or veterinary use.

Target PI3K
Research area Cancer
Purity >98% Stock Inquire

Gilmelisib structure

CAS No.: 1845777-61-8

Download structure (.mol)

Pack sizes & pricing

Size Price SKU Stock
10 mg USD 550.00 BP-02232-10mg In stock Get quote
25 mg USD 885.00 BP-02232-25mg In stock Get quote
50 mg USD 1,285.00 BP-02232-50mg In stock Get quote
100 mg USD 1,885.00 BP-02232-100mg In stock Get quote
250 mg USD 2,885.00 BP-02232-250mg In stock Get quote
500 mg USD 3,980.00 BP-02232-500mg In stock Get quote

Need another size or custom synthesis? Request a quote.

Description

Gilmelisib is an antineoplastic. Gilmelisib is a PI3K inhibitor (IC50 <1 nM for PI3K p110α) extracted from WO2017101847 A1, compound 1.

Biological activity

Gilmelisib is an antineoplastic. Gilmelisib is a PI3K inhibitor (IC50 <1 nM for PI3K p110α).

Specifications

MW (average)
547.9860
Formula
C24H23ClFN5O5S
CAS No.
1845777-61-8
Physical state
Solid
Color
White to yellow
Shipping
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage
Powder -20℃ 3 years; In solvent -20℃ 1 month;

Solubility

DMSO 5 mg/mL (ultrasonic and warming and adjust pH to 4 with HCl and heat to 60°C)

References

[1]. WO2017101847 A1
[2]. International Nonproprietary Names for Pharmaceutical Substances (INN)

Same target

Search PI3K

Same research area

Search Cancer